Available
$58.00
Strict Regulatory Notice: This agent is synthesized strictly for laboratory-based research and analytical purposes. It is not intended for human or veterinary use, nor for medical, household, or cosmetic applications. Please review our Terms of Service thoroughly before finalizing your acquisition.
25mg/mL solution (750mg/30mL)
25mg/mL Oil (500mg/20mL)
| Parameter | Specification / Details |
|---|---|
| Primary Compound Name | GW501516 (PPARδ Agonist) |
| CAS Registry Number | 317318-70-0 |
| IUPAC Designation | 2-[2-methyl-4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenoxy]acetic acid |
| Synonyms / Trade Names | Cardarine, Endurobol, GSK-516 |
| PubChem CID | 9803963 |
| Molecular Formula | C₂₁H₁₈F₃NO₃S₂ |
| Molar Mass / Weight | 453.50 g/mol |
| Physical Appearance | White to off-white crystalline powder (raw) / Clear or slightly tinted liquid (suspended) |
| Solubility Profile | Soluble in DMSO, Ethanol, and Propylene Glycol/PEG 400. Insoluble in water. |
| Tested Purity | ≥99% via HPLC |
| Active Ingredient (Total) | 600mg per 30mL vial |
| Dry / Powder Formulations | N/A (Liquid suspension) |
| Liquid / Solution Concentrations | 20mg/mL in a PEG 400 / Ethanol carrier |
| Alternative Formulations | GW0742 (Fitorine - a closely related PPARδ agonist) |
| Storage Guidelines | Store at room temperature (20°C to 25°C). Protect strictly from moisture, heat, and direct sunlight. |
| Estimated Shelf Life | 24 months from manufacture date. |
| Safety Documentation | Standard SDS available for GW501516 |
| Terms of Application | For laboratory research purposes only. Not for human or veterinary use. Investigated for its role as a high-affinity PPARδ agonist to evaluate fatty acid oxidation, mitochondrial biogenesis, and metabolic signaling in in-vitro models. |
GW501516 (Cardarine) is a paramount subject within the field of cellular bioenergetics and exercise mimetic pharmacology. As a highly potent peroxisome proliferator-activated receptor delta (PPARδ) agonist, it has become a staple for researchers examining the shift from glucose oxidation to lipid oxidation, mitochondrial biogenesis, and skeletal muscle fiber type switching.
At 4 Amino Labs, we provide this complex in a highly purified format to ensure experimental reproducibility. By maintaining rigorous measurement standards, we provide the consistency required for longitudinal data integrity.
Scientific Literature Reference: The biochemical pathway of PPARδ acting as an “exercise mimetic” by fundamentally altering fuel preference at the mitochondrial level is a cornerstone of modern metabolic research. See: Narkar, V. A., et al. (2008). “AMPK and PPARdelta agonists are exercise mimetics.” Cell, 134(3), 405-415.
Our GW501516 undergoes a multifaceted verification process. Each batch is subjected to independent High-Performance Liquid Chromatography (HPLC) to ensure a purity threshold of ≥ 99%. This analytical rigor ensures the absence of cross-contaminants or heavy metal degradation products.
Researchers utilizing GW501516 typically focus on the following biochemical mechanisms:
To maintain the molecular integrity of GW501516, the following storage parameters are recommended:
This substance is provided exclusively for in-vitro laboratory research and pre-clinical developmental testing. 4 Amino Lab does not condone or authorize the use of this product in any clinical setting or for personal consumption. Misuse of laboratory chemicals carries significant health risks. By purchasing, the researcher acknowledges the inherent risks and confirms they possess the necessary equipment and expertise to handle these materials safely.
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